Fig. 1 · Structure
Documents & Downloads
Rupatadine-d4 fumarate
Deuterated Rupatadine Fumarate
Rupatadine-d4 fumarate is a deuterated derivative of Rupatadine fumarate, targeting dual platelet-activating factor (PAF) and H1 receptors. It demonstrates potent antagonistic activity, with Ki values of 0.55 μM for PAF and 0.1 μM for the H1 receptor, making it a valuable tool for studies of allergic reactions and inflammatory processes. This reagent is particularly useful in pharmacological research exploring the modulation of allergic responses and related signaling pathways.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 1795153-63-7 |
| Applications | Deuterated Rupatadine Fumarate |
| Formula | C30H26D4ClN3O4 |
| Molecular Weight | 536.05 |
| Synonyms | UR-12592 D4 fumarate |
| SMILES | CC1=CN=CC(CN2C([2H])([2H])C/C(CC2([2H])[2H])=C3C4=CC=C(Cl)C=C4CCC5=CC=CN=C5\3)=C1.OC(/C=C/C(O)=O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.