RVX-208

Catalog No.: A13956

BET bromodomain inhibitor

RVX-208

RVX-208 Chemical Structure

CAS NO. 1044870-39-4

RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 uM for BD2, about 170-fold selectivity over BD1.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $100.00

Special Price $90.00

25 mg

Regular Price: $200.00

Special Price $180.00

50 mg

Regular Price: $350.00

Special Price $315.00

10mM * 1mL in DMSO

Regular Price: $75.00

Special Price $67.50

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 uM for BD2, about 170-fold selectivity over BD1.
Targets
BD2 (Cell-free assay)
0.51 μM
In vitro DMSO 74 mg/mL (199.78 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27 mL 134.99 mL 269.98 mL
0.5 mM 5.4 mL 27 mL 54 mL
1 mM 2.7 mL 13.5 mL 27 mL
5 mM 0.54 mL 2.7 mL 5.4 mL

*The above data is based on the productmolecular weight 370.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13956
Actions Inhibitor
M. Wt 370.4
Formula C20H22N2O5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1044870-39-4
Synonyms RVX-000222
SMILES CC1=CC(=CC(=C1OCCO)C)C2=NC(=O)C3=C(C=C(C=C3N2)OC)OC

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy RVX-208 | RVX-208 Supplier | purchase RVX-208 | RVX-208 cost | RVX-208 manufacturer | order RVX-208 | RVX-208 distributor | buy 1044870-39-4| 1044870-39-4 Supplier | purchase 1044870-39-4 | 1044870-39-4 cost | 1044870-39-4 manufacturer | order 1044870-39-4 | 1044870-39-4 distributor
Rewards