Fig. 1 · Structure
Documents & Downloads
(S,S)-CPI-1612
Isomer
(S,S)-CPI-1612 is an isomer of the potent EP300/CBP histone acetyltransferase (HAT) inhibitor CPI-1612, exhibiting an IC50 of 8.1 nM for EP300 HAT. As an experimental control, (S,S)-CPI-1612 is essential for validating the biological effects of its counterpart, particularly in cancer research. This compound facilitates investigations into the role of histone acetylation in cancer progression and treatment responses.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2374971-82-9 |
| Applications | Isomer |
| Formula | C27H26N6O |
| Molecular Weight | 450.53 |
| SMILES | CN(N=C1)C=C1C(C=N2)=CC=C2NC([C@H](C3=CC=CC=C3)NC[C@H](C4=CC=C(C=C4)C#N)C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.