Fig. 1 · Structure
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S6821
TAS2R8 Antagonist
S6821 is a potent antagonist of the TAS2R8 receptor, exhibiting an IC50 value of 0.035 μM. This compound demonstrates a favorable safety profile, as it has not exhibited mutagenic properties in vitro and does not induce micronucleus formation in bone marrow polychromatic erythrocytes in vivo. S6821 is suitable for research applications involving taste signaling pathways and receptor pharmacology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1119831-25-2 |
| Applications | TAS2R8 Antagonist |
| Formula | C19H19N5O4 |
| Molecular Weight | 381.39 |
| SMILES | O=C1N(C2=CN(CC3=C(C)ON=C3C)N=C2)C(CN1CC4=CC(O)=CC=C4)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.