Samidorphan is an opioid receptor modulator with a high affinity for μ-opioid, κ-opioid, and δ-opioid receptors. It functions as an antagonist at μ-opioid receptors while serving as a partial agonist at κ- and δ-opioid receptors. This unique profile allows Samidorphan to primarily act as an opioid antagonist in vivo, demonstrating potential for improving depressive behaviors in animal models. Its mechanistic action makes it a valuable tool for research in the fields of pain management, addiction, and mood disorders.
Samidorphan is an opioid receptor modulator with a high affinity for μ-opioid, κ-opioid, and δ-opioid receptors. It functions as an antagonist at μ-opioid receptors while serving as a partial agonist at κ- and δ-opioid receptors. This unique profile allows Samidorphan to primarily act as an opioid antagonist in vivo, demonstrating potential for improving depressive behaviors in animal models. Its mechanistic action makes it a valuable tool for research in the fields of pain management, addiction, and mood disorders.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
