• Sign In
  • FAQ
  • Create an Account
Currency
USD currency flagUSD
Toggle Nav
My Cart
Menu
Account
Settings
Currency
USD currency flagUSD

SC-53606

Catalog No.: A29612
5-HT4 Receptor Antagonist
SC-53606 is a potent and selective antagonist of the 5-HT4 receptor, exhibiting a pA2 value of 8.13. It effectively inhibits the 5-HT4 receptor-mediated relaxation in Carbachol-induced contractions, making it valuable for studying gastrointestinal motility and related disorders. This compound is useful in research focused on neuropharmacology and the serotonergic system.
SC-53606 151898-33-8 5-HT4 Receptor Antagonist
Grouped product items
Size Price Stock Qty
25mg
$1,405.00
In stock
50mg
$1,790.00
In stock
100mg
$2,240.00
In stock
Bulk Size
Bulk Discount
Bulk Inquiry
Notify me when the price drops
Free Delivery on orders over $500
Research use only. We do not sell to patients.
Data Sheet SDS

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionSC-53606 is a potent and selective antagonist of the 5-HT4 receptor, exhibiting a pA2 value of 8.13. It effectively inhibits the 5-HT4 receptor-mediated relaxation in Carbachol-induced contractions, making it valuable for studying gastrointestinal motility and related disorders. This compound is useful in research focused on neuropharmacology and the serotonergic system.
Product Information
Catalog NumA29612
FormulaC16H19ClN4O
Molecular Weight318.80
CAS Number151898-33-8
SMILESO=C(NC[C@H]1[C@@]2(CCCN2CC1)[H])C3=CC(Cl)=CN4C3=NC=C4
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

GPCR/G Protein > 5-HT Receptors