Fig. 1 · Structure
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SENP2-IN-1
SENP2 Inhibitor
SENP2-IN-1 is a selective SENP2 inhibitor, targeting the SUMO-specific protease SENP2 with potent inhibitory activity. It demonstrates IC50 values of 1.3 μM for SENP1, 0.69 μM for SENP2, and 22.7 μM for SENP5, indicating a strong selectivity towards SENP2. This compound is valuable for cancer research, providing insights into the role of SENP2 in tumor biology and potential therapeutic developments.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2986220-46-4 |
| Applications | SENP2 Inhibitor |
| Formula | C32H29N3O5S2 |
| Molecular Weight | 599.72 |
| SMILES | O=C(OCC)CNC1=CC=C2C(C(OCC3=CC=CC=C3)=C(C(NCC4=CC=CC(NC(C5=CC=CS5)=O)=C4)=O)S2)=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.