Fig. 1 · Structure
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Setin-1
Set7 Inhibitor
Setin-1 is a potent inhibitor of Set7, functioning as a lysine methyltransferase (KMTase) inhibitor. It effectively impedes the enzymatic activity of Set7, influencing the methylation status of histones and non-histone proteins. This compound is valuable for research applications involving epigenetic regulation, cellular differentiation, and gene expression studies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1313802-67-3 |
| Applications | Set7 Inhibitor |
| Formula | C29H21F3N2O2 |
| Molecular Weight | 486.48 |
| SMILES | FC(F)(C1=CC=C(C=C1)C2=CC=CC3=C2C=CN3C4=CC(CNC5=CC(C(O)=O)=CC=C5)=CC=C4)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.