SP2509 (HCI-2509)
Important Notice: For research use only. We do not sell to patients.
Loading distributor info...
Important Notice: For research use only. We do not sell to patients.
Loading distributor info...
Discription | SP2509 is a novel histone demethylase LSD1 (KDM1A) antagonist with IC50 of 13 nM; no inhibition on MAO-A and MAO-B. | ||
---|---|---|---|
Targets |
|
Catalog Num | A14443 |
---|---|
Formula | C19H20ClN3O5S |
Molecular Weight | 437.9 |
CAS Number | 1423715-09-6 |
SMILES | CC(=C1C=C(C=CC1=O)Cl)NNC(=O)C2=CC(=CC=C2)S(=O)(=O)N3CCOCC3 |
Synonyms | SP-2509 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 36 mg/mL (82.2 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 10% DMSO+corn oil | 4 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.84 mL | 114.18 mL | 228.36 mL |
0.5 mM | 4.57 mL | 22.84 mL | 45.67 mL |
1 mM | 2.28 mL | 11.42 mL | 22.84 mL |
5 mM | 0.46 mL | 2.28 mL | 4.57 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2