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$0.00 - Ming Tang, .et al. Celastrol alleviates renal fibrosis by upregulating cannabinoid receptor 2 expression, Cell Death Dis, 2018, Jun; 9(6): 601 PMID: 29789558
Biological Activity
SR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.01 mL | 105.03 mL | 210.06 mL |
| 0.5 mM | 4.2 mL | 21.01 mL | 42.01 mL |
| 1 mM | 2.1 mL | 10.5 mL | 21.01 mL |
| 5 mM | 0.42 mL | 2.1 mL | 4.2 mL |
*The above data is based on the productmolecular weight 476.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A12376 |
|---|---|
| Actions | Agonist |
| M. Wt | 476.05 |
| Formula | C29H34ClN3O |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 192703-06-3 |
| Synonyms | SR144528, SR-144528 |
| SMILES | CC1=CC=C(C=C1)CN2C(=CC(=N2)C(=O)N[[email protected]]3[[email protected]]4(CC[[email protected]](C4)C3(C)C)C)C5=CC(=C(C=C5)Cl)C |
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