SR 144528

Catalog No.: A12376

CB2 inverse agonist

SR 144528

SR 144528 Chemical Structure

CAS NO. 192703-06-3

SR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors.

Availability: In stock

Package Price Qty
5 mg
$95.00
10 mg
$170.00
25 mg
$390.00
50 mg
$670.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Ming Tang, .et al. Celastrol alleviates renal fibrosis by upregulating cannabinoid receptor 2 expression, Cell Death Dis, 2018, Jun; 9(6): 601 PMID: 29789558

Biological Activity

SR 144528 is a selective peripheral cannabinoid receptor inverse agonist that displays a Ki value of 0.6 nM for rat spleen and human recombinant CB2 receptors and a Ki value of 400 nM for rat brain and human recombinant CB1 receptors.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.01 mL 105.03 mL 210.06 mL
0.5 mM 4.2 mL 21.01 mL 42.01 mL
1 mM 2.1 mL 10.5 mL 21.01 mL
5 mM 0.42 mL 2.1 mL 4.2 mL

*The above data is based on the productmolecular weight 476.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12376
Actions Agonist
M. Wt 476.05
Formula C29H34ClN3O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 192703-06-3
Synonyms SR144528, SR-144528
SMILES CC1=CC=C(C=C1)CN2C(=CC(=N2)C(=O)N[[email protected]]3[[email protected]]4(CC[[email protected]](C4)C3(C)C)C)C5=CC(=C(C=C5)Cl)C

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