Fig. 1 · Structure
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TAI-1
Hec1 Inhibitor
TAI-1 is a potent inhibitor of Hec1, demonstrating a GI50 of 13.48 nM in K562 cells. This orally active anticancer agent offers significant potential for the treatment of cancers associated with Hec1 dysregulation. TAI-1 is valuable for research applications focused on elucidating the role of Hec1 in tumorigenesis and exploring targeted therapeutic strategies in oncology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1334921-03-7 |
| Applications | Hec1 Inhibitor |
| Formula | C24H21N3O3S |
| Molecular Weight | 431.51 |
| SMILES | O=C(C1=CC=NC=C1)NC2=NC(C3=C(C)C=C(OC4=CC=C(OC)C=C4)C=C3C)=CS2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.