Fig. 1 · Structure
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TAK-448
KISS1R Agonist
TAK-448 is a potent and selective agonist for the KISS1 receptor (KISS1R), exhibiting an IC50 of 460 pM and an EC50 of 632 pM. This compound significantly stimulates KISS1R activity, making it valuable for research into reproductive biology and related signaling pathways. Its use can provide insights into the role of KISS1R in various physiological processes, including hormone regulation and metastasis.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 1234319-68-6 |
| Applications | KISS1R Agonist |
| Formula | C58H80N16O14 |
| Molecular Weight | 1225.36 |
| Synonyms | MVT-602 |
| SMILES | C([C@H](NC([C@@H](NC([C@@H](NC(NNC([C@H](CC1=CC=CC=C1)NC([C@@H](NC([C@@H](NC(=O)[C@H]2N(C([C@@H](CC3=CC=C(O)C=C3)NC(C)=O)=O)C[C@H](O)C2)CC(N)=O)=O)[C@@H](C)O)=O)=O)=O)CC(C)C)=O)CCCNC(NC)=N)=O)C(N)=O)C=4C=5C(NC4)=CC=CC5 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.