TAK-981

Catalog No.: A20002

SUMO inhibitor

TAK-981

TAK-981 Chemical Structure

CAS NO. 1858276-04-6

TAK-981 is a first in class and selective inhibitor of the SUMOylation enzymatic cascade, with potential immune-activating and antineoplastic activities.

Availability: In stock

Package Price Qty
1 mg
$320.00
5 mg
$960.00
10 mg
$1,600.00
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Biological Activity

TAK-981 is a first in class and selective inhibitor of the SUMOylation enzymatic cascade, with potential immune-activating and antineoplastic activities.
In vitro DMSO 97 mg/mL (167.79 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.3 mL 86.49 mL 172.98 mL
0.5 mM 3.46 mL 17.3 mL 34.6 mL
1 mM 1.73 mL 8.65 mL 17.3 mL
5 mM 0.35 mL 1.73 mL 3.46 mL

*The above data is based on the productmolecular weight 578.1. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20002
Actions Inhibitor
CAS No. 1858276-04-6
Formula C25H28ClN5O5S2
M. Wt 578.1
Purity >98%
Synonyms TAK981, TAK 981
SMILES O=S(OC[[email protected]@H]1[[email protected]@H](O)C[[email protected]](NC2=NC=NC=C2C(C3=CC([[email protected]@H]4NCCC5=C4C=C(Cl)C=C5)=C(C)S3)=O)C1)(N)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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