TAS-116

Catalog No.: A20987

HSP90α/HSP90β inhibitor

TAS-116

TAS-116 Chemical Structure

CAS NO. 1260533-36-5

TAS-116 is an oral bioavailable, ATP-competitive, highly specific HSP90α/HSP90β inhibitor (Kis of 34.7 nM and 21.3 nM, respectively) without inhibiting other HSP90 family proteins such as GRP94. TAS-116 demonstrates less ocular toxicity.

Availability: In stock

Package Price Qty
5 mg
$77.00
10 mg
$132.00
50 mg
$391.00
100 mg
$782.00
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Biological Activity

TAS-116 is an oral bioavailable, ATP-competitive, highly specific HSP90α/HSP90β inhibitor (Kis of 34.7 nM and 21.3 nM, respectively) without inhibiting other HSP90 family proteins such as GRP94. TAS-116 demonstrates less ocular toxicity.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22 mL 110 mL 220.01 mL
0.5 mM 4.4 mL 22 mL 44 mL
1 mM 2.2 mL 11 mL 22 mL
5 mM 0.44 mL 2.2 mL 4.4 mL

*The above data is based on the productmolecular weight 454.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20987
Actions Inhibitor
M. Wt 454.53
Formula C25H26N8O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1260533-36-5
Synonyms TAS116, TAS 116
SMILES O=C(N)C1=CC=C(N2N=C(C(C)C)C3=C(N4C=C(C5=CN(C)N=C5)N=C4)C=CN=C32)C(CC)=C1

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