Tebapivat

Catalog No.: A77400
Pyruvate Kinase-R Activator
Tebapivat is a potent activator of pyruvate kinase-R (PKR), playing a critical role in enhancing glycolytic flux and energy metabolism. Its ability to stimulate PKR makes it valuable in research on metabolic disorders and cancer, where glycolysis is often dysregulated. Tebapivat can be utilized to investigate the effects of PKR activation on cellular energy production and related biochemical pathways.
Grouped product items
Size Price Stock Qty
1mg
$720.00
In stock
5mg
$960.00
In stock
10mg
$1,100.00
In stock
25mg
$1,275.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionTebapivat is a potent activator of pyruvate kinase-R (PKR), playing a critical role in enhancing glycolytic flux and energy metabolism. Its ability to stimulate PKR makes it valuable in research on metabolic disorders and cancer, where glycolysis is often dysregulated. Tebapivat can be utilized to investigate the effects of PKR activation on cellular energy production and related biochemical pathways.
Product Information
Catalog NumA77400
FormulaC18H16N8OS
Molecular Weight392.44
CAS Number2283422-04-6
SMILESO=C1C(N(C)C2=C3SC(CC4=NNC=C4)=N2)=C3C=NN1CC5=NC(N)=CC=C5
SynonymsAG-946; PKR activator 2
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2