Fig. 1 · Structure
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Telmisartan-13C,d3
Stable Isotope
Telmisartan-13C,d3 is a stable isotope-labeled version of Telmisartan, a potent and long-acting antagonist of the angiotensin II type 1 receptor (AT1). It selectively inhibits the binding of 125I-AngII to AT1 receptors, exhibiting an IC50 value of 9.2 nM. This reagent is valuable for pharmacological studies and metabolic research, particularly in tracking drug metabolism and pharmacokinetics in biological systems.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 1261396-33-1 |
| Applications | Stable Isotope |
| Formula | C3213CH27D3N4O2 |
| Molecular Weight | 518.63 |
| Synonyms | BIBR 277-13C,d3 |
| SMILES | CCCC(N(C1=CC(C2=NC3=CC=CC=C3N2[13C]([2H])([2H])[2H])=C4)CC5=CC=C(C6=C(C=CC=C6)C(O)=O)C=C5)=NC1=C4C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.