Fig. 1 · Structure
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Telmisartan-d3
Stable Isotope
Telmisartan-d3 is a deuterium-labeled derivative of Telmisartan, a potent and long-lasting antagonist of the angiotensin II type 1 receptor (AT1). This compound selectively inhibits the binding of 125I-AngII to AT1 receptors, exhibiting an IC50 value of 9.2 nM. Telmisartan-d3 serves as a valuable stable isotope for pharmacokinetic studies and in investigations involving the modulation of blood pressure and related cardiovascular research.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 1189889-44-8 |
| Applications | Stable Isotope |
| Formula | C33H27D3N4O2 |
| Molecular Weight | 517.64 |
| SMILES | CC1=CC(C2=NC3=C(N2C([2H])([2H])[2H])C=CC=C3)=CC4=C1N=C(N4CC5=CC=C(C=C5)C6=CC=CC=C6C(O)=O)CCC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.