Fig. 1 · Structure
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Thioperamide maleate
H3 Antagonist
Thioperamide maleate is a selective H3 receptor antagonist known for its ability to inhibit [3H]histamine release with a Ki of 4.3 nM. This compound effectively interferes with [3H]histamine synthesis, exhibiting a Ki of 31 nM. Thioperamide maleate is primarily used in neurological research to study histamine signaling and its implications in various physiological and pathological conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 148440-81-7 |
| Applications | H3 Antagonist |
| Formula | C15H24N4S.xC4H4O4 |
| Molecular Weight | 408.52 |
| Synonyms | MR-12842 maleate |
| SMILES | S=C(N1CCC(C2=CN=CN2)CC1)NC3CCCCC3.O=C(O)/C=C\C(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.