Target & Activity
| Target | Activity | Value |
|---|---|---|
| LTD4 | 6.41 (pA2, In guinea-pigs) | |
| LTE4 | 6.45 (pA2, In guinea-pigs) |
Fig. 1 · Structure
Documents & Downloads
Tipelukast
Cat. No.
A21249
CAS
125961-82-2
leukotriene receptor antagonist
Tipelukast (KCA 757) is a sulfidopeptide leukotriene receptor antagonist, an orally bioavailable anti-inflammatory agent and used for the treatment of asthma.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Biological Activity
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 125961-82-2 |
| Applications | leukotriene receptor antagonist |
| Formula | C29H38O7S |
| Molecular Weight | 530.67 |
| Synonyms | KCA 757; MN 001 |
| SMILES | CC(C1=C(O)C(CCC)=C(SCCCOC2=C(CCC)C(OCCCC(O)=O)=C(C(C)=O)C=C2)C=C1)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.