Fig. 1 · Structure
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(+)-TK216 (d-TK216)
TK216 Enantiomer
(+)-TK216 is the active enantiomer of TK216, serving as a potent inhibitor of the E26 transformation specific (ETS) transcription factors. This compound exhibits significant biological activity in modulating gene expression and has shown promise in cancer research due to its ability to disrupt ETS-related signaling pathways. It is a valuable reagent for investigating the role of ETS proteins in oncogenesis and other related cellular processes.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1903783-77-6 |
| Applications | TK216 Enantiomer |
| Formula | C19H15Cl2NO3 |
| Molecular Weight | 376.23 |
| Synonyms | d-TK216 |
| SMILES | O=C1NC2=C(C(Cl)=CC=C2Cl)C1(CC(C3=CC=C(C4CC4)C=C3)=O)O.[Rotation (+)] |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.