TLK117

Catalog No.: A21531

TLK117

TLK117 Chemical Structure

CAS NO. 152684-53-2

TLK117, the active metabolite of TLK199, selective inhibits Glutathione S-transferase P1?C1 (GSTP1-1) with a Ki of 0.4 μM for GSTP. TLK117 also competitively inhibits glyoxalase I with a Ki of 0.56 μM.

Availability: In stock

Package Price Qty
5 mg
$162.00
10 mg
$279.00
50 mg
$828.00
100 mg
$1,656.00
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Biological Activity

TLK117, the active metabolite of TLK199, selective inhibits Glutathione S-transferase P1?C1 (GSTP1-1) with a Ki of 0.4 μM for GSTP. TLK117 also competitively inhibits glyoxalase I with a Ki of 0.56 μM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.12 mL 105.59 mL 211.18 mL
0.5 mM 4.22 mL 21.12 mL 42.24 mL
1 mM 2.11 mL 10.56 mL 21.12 mL
5 mM 0.42 mL 2.11 mL 4.22 mL

*The above data is based on the productmolecular weight 473.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21531
CAS No. 152684-53-2
Formula C23H27N3O6S
M. Wt 473.54
Purity >98%
Synonyms TLK-117, TLK 117, TER117, TER-117, TER 117
SMILES O=C(O)[[email protected]@H](C1=CC=CC=C1)NC([[email protected]@H](NC(CC[[email protected]](N)C(O)=O)=O)CSCC2=CC=CC=C2)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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