Fig. 1 · Structure
Documents & Downloads
Tolvaptan-d7
Stable Isotope
Tolvaptan-d7 is a deuterium-labeled variant of Tolvaptan, a selective antagonist of arginine vasopressin receptor 2 (AVPR2). This compound exhibits an IC50 of 1.28 μM in inhibiting AVP-induced platelet aggregation. Tolvaptan-d7 is utilized in biological research for studying the pharmacokinetics and metabolic pathways of Tolvaptan, providing insights into its therapeutic effects and mechanisms of action.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 1246818-18-7 |
| Applications | Stable Isotope |
| Formula | C26H18D7ClN2O3 |
| Molecular Weight | 455.98 |
| SMILES | O=C(C1=C(C=C(C=C1)NC(C2=C(C([2H])=C([2H])C([2H])=C2[2H])C([2H])([2H])[2H])=O)C)N3C4=CC=C(Cl)C=C4C(CCC3)O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.