Fig. 1 · Structure
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TP-5801
TNK1 Inhibitor
TP-5801 is a potent inhibitor of TNK1 (non-receptor tyrosine kinase), demonstrating an IC50 value of 1.40 nM. This compound exhibits significant anti-tumor activity, making it a valuable tool for cancer research. Its selective inhibition of TNK1 may provide insights into oncogenic signaling pathways and therapeutic strategies for targeting malignancies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2574474-81-8 |
| Applications | TNK1 Inhibitor |
| Formula | C24H31BrN8O |
| Molecular Weight | 527.46 |
| SMILES | CN1CCN(C2=C(C)C=C(NC3=NC=C(Br)C(NC4=CC=CN=C4N(C)C)=N3)C(OC)=C2)CC1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.