Fig. 1 · Structure
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TRIM24/BRPF1-IN-2
TRIM24/BRPF1 Inhibitor
TRIM24/BRPF1-IN-2 is a dual inhibitor targeting TRIM24 and BRPF1, exhibiting IC50 values of 0.98 μM and 1.16 μM, respectively. This compound demonstrates strong binding affinity to the bromodomains of TRIM24 and BRPF1. TRIM24/BRPF1-IN-2 is particularly relevant for research into prostate cancer, providing a valuable tool for understanding the role of these proteins in tumorigenesis.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 3033288-68-2 |
| Applications | TRIM24/BRPF1 Inhibitor |
| Formula | C20H22N2O4S |
| Molecular Weight | 386.46 |
| SMILES | COC1=CC=C(C=C1S(=O)(NC2=CC=C3C(CCN3C(C)=O)=C2)=O)C4CC4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.