Fig. 1 · Structure
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UNC0737
Orthosteric Choline Kinase Inhibitor
UNC0737 is an orthosteric choline kinase inhibitor that selectively targets choline kinase with significant potency. This compound exhibits limited inhibition of G9a and GLP, with IC50 values of 5000 nM and greater than 10000 nM, respectively, as determined in SAHH-coupled assays. UNC0737 is valuable for research applications investigating choline metabolism and its implications in various cellular processes and diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1327276-39-0 |
| Applications | Orthosteric Choline Kinase Inhibitor |
| Formula | C31H49N5O2 |
| Molecular Weight | 523.75 |
| SMILES | CN(C1CCN(C(C)C)CC1)C2=NC(C3CCCCC3)=NC4=C2C=C(OC)C(OCCCN5CCCC5)=C4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.