Fig. 1 · Structure
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Usmarapride free base
5-HT4 Receptor Agonist
Usmarapride free base is a selective partial agonist of the 5-HT4 receptor, exhibiting a potent activity with an EC50 of 44 nM. This compound is orally active and can penetrate the blood-brain barrier, making it suitable for investigations into cognitive deficits related to Alzheimer's disease. Its mechanism of action supports research aimed at understanding and potentially mitigating Alzheimer's-associated cognitive impairments.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Partial Agonist |
| CAS Number | 1428862-32-1 |
| Applications | 5-HT4 Receptor Agonist |
| Formula | C21H29N5O2 |
| Molecular Weight | 383.49 |
| Synonyms | SUVN-D4010 free base |
| SMILES | CC(N1N=C(C2=NN=C(C3CCN(CCCOC)CC3)O2)C4=C1C=CC=C4)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.