Fig. 1 · Structure
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Usmarapride
5-HT4 Receptor Agonist
Usmarapride is a selective agonist of the 5-HT4 receptor, exhibiting potent activity with an EC50 of 27.5 nM. This compound is orally active and demonstrates the ability to penetrate the blood-brain barrier, making it a valuable tool for investigating cognitive deficits related to Alzheimer's disease. Usmarapride is primarily utilized in research focused on neuropsychological disorders and related therapeutic strategies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 1428862-33-2 |
| Applications | 5-HT4 Receptor Agonist |
| Formula | C23H31N5O6 |
| Molecular Weight | 473.52 |
| Synonyms | SUVN-D4010 |
| SMILES | CC(N1N=C(C2=NN=C(C3CCN(CCCOC)CC3)O2)C4=C1C=CC=C4)C.O=C(O)C(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.