Fig. 1 · Structure
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VA-111913
Vasopressin Receptor V1A Antagonist
VA-111913 is a potent antagonist of the vasopressin receptor V1A, exhibiting a Ki value of 1.74 nM. This compound has demonstrated efficacy in reducing uterine contractions and enhancing uterine blood flow through the inhibition of vasopressin, making it relevant for studies focused on alleviating dysmenorrhea. VA-111913 serves as a valuable tool for research on menstrual pain and its associated mechanisms.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 877856-17-2 |
| Applications | Vasopressin Receptor V1A Antagonist |
| Formula | C23H21ClFN5O2 |
| Molecular Weight | 453.90 |
| Synonyms | VT-913 |
| SMILES | O=C(C1CC1)NCC2=CC=C(C(N3CC4=C(N(C)N=C4)NC5=CC(Cl)=CC=C35)=O)C=C2F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.