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VAP-1-IN-2

VAP-1 Inhibitor

VAP-1-IN-2 is a potent oral inhibitor of VAP-1, demonstrating an IC50 of 0.025 μM against human VAP-1 and 0.015 μM against rat VAP-1. This compound effectively reduces urinary protein excretion and mitigates the progression of proteinuria in diabetic rat models. VAP-1-IN-2 is valuable for research focused on diabetes and nephropathy mechanisms.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	1279026-89-9
Applications	VAP-1 Inhibitor
Formula	C₂₅H₂₇ClN₆O₃
Molecular Weight	494.98
SMILES	O=C(O)C1=CC=C(C(Cl)=C1)N2CCN(C=3N=CC(=CN3)C4=CC=CC(=C4)CN(C(=O)CN)C)CC2

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.