Fig. 1 · Structure
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Vasopressin V2 receptor antagonist 1
V2R Antagonist
Vasopressin V2 receptor antagonist 1 functions as a selective antagonist of the vasopressin V2 receptor (V2R) with a Ki value of 3.8 nM. This compound is primarily utilized in research focusing on autosomal dominant polycystic kidney disease (ADPKD) and has potential implications in studying renal pathophysiology and therapeutics. Its specificity for V2R makes it a valuable tool for elucidating the receptor's role in kidney function and associated disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2648650-50-2 |
| Applications | V2R Antagonist |
| Formula | C33H37ClN4O4 |
| Molecular Weight | 589.12 |
| SMILES | ClC1=CC2=C(C=C1)N(C(C3=C(C=C(C=C3)NC(C4=C(C=CC=C4)C)=O)C)=O)CCCC2NCCC(N5CCOCC5)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.