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Velmupressin

V2R Agonist

Velmupressin is a potent and selective peptidic agonist of the V2 receptor (V2R), with effective concentrations (EC50) of 0.07 nM for human V2R and 0.02 nM for rat V2R. This short-acting compound is utilized in research applications focusing on water conservation and aquaporin regulation, providing valuable insights into renal physiology and potential therapeutic interventions in conditions such as diabetes insipidus.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Agonist
CAS Number	1647119-61-6
Applications	V2R Agonist
Formula	C₄₂H₆₀ClN₁₁O₈S₂
Molecular Weight	946.58
Synonyms	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
SMILES	C(=O)(N1[C@H](C(NCCCCNC(=N)N)=O)CCC1)[C@H]2NC(=O)[C@H](CC(N)=O)NC(=O)[C@H]([C@@H](C)C)NC(=O)[C@H](CC3=CC=CS3)NC(=O)[C@H](CC4=CC=C(Cl)C=C4)NC(=O)CCCSC2

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.