Fig. 1 · Structure
Documents & Downloads
Velusetrag
5-HT4R Agonist
Velusetrag is a potent and selective agonist of the serotonin 5-HT4 receptor (5-HT4R), demonstrating a pKi of 7.7. It exhibits minimal affinity for 5-HT2A and 5-HT2B receptors, ensuring a specific receptor interaction. This compound is primarily utilized in research related to gastrointestinal disorders and Parkinson's disease, contributing to the understanding of serotonergic modulation in these conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 866933-46-2 |
| Applications | 5-HT4R Agonist |
| Formula | C25H36N4O5S |
| Molecular Weight | 504.64 |
| Synonyms | TD-5108 |
| SMILES | O=C(C1=CC2=C(N(C(C)C)C1=O)C=CC=C2)N[C@@H]3C[C@@H](N4C[C@@H](O)CN(C)S(=O)(C)=O)CC[C@@H]4C3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.