VU0530244 is a highly potent antagonist of the serotonin 5-HT2B receptor, exhibiting an IC50 of 17.3 nM. Due to its predicted properties, VU0530244 is expected to have minimal brain penetration in human subjects and is likely a substrate for P-glycoprotein-mediated efflux. This compound is useful for research applications focused on serotonin receptor signaling and its implications in various physiological and pathological processes.
VU0530244 is a highly potent antagonist of the serotonin 5-HT2B receptor, exhibiting an IC50 of 17.3 nM. Due to its predicted properties, VU0530244 is expected to have minimal brain penetration in human subjects and is likely a substrate for P-glycoprotein-mediated efflux. This compound is useful for research applications focused on serotonin receptor signaling and its implications in various physiological and pathological processes.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
