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WEHI-539 hydrochloride is a small-molecule inhibitor of BCL-xL with IC50 value of 1.1 nM.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 16.12 mL | 80.62 mL | 161.24 mL |
| 0.5 mM | 3.22 mL | 16.12 mL | 32.25 mL |
| 1 mM | 1.61 mL | 8.06 mL | 16.12 mL |
| 5 mM | 0.32 mL | 1.61 mL | 3.22 mL |
*The above data is based on the productmolecular weight 620.18. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13327 |
|---|---|
| Actions | Inhibitor |
| CAS No. | Not avalable. |
| Formula | C31H30ClN5O3S2 |
| M. Wt | 620.18 |
| Solubility | DMSO |
| Purity | >98% |
| Synonyms | WEHI539 hydrochloride, WEHI 539 hydrochloride |
| SMILES | O=C(C1=C(C([H])([H])C([H])([H])C([H])([H])OC2=C([H])C([H])=C(C([H])([H])N([H])[H])C([H])=C2[H])SC(C3=C([H])C4=C(C([H])=C3[H])C([H])([H])C([H])([H])C([H])([H])/C4=N\N([H])C5=NC6=C([H])C([H])=C([H])C([H])=C6S5)=N1)O[H] |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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