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Biological Activity
WEHI-539 hydrochloride is a small-molecule inhibitor of BCL-xL with IC50 value of 1.1 nM.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 16.12 mL | 80.62 mL | 161.24 mL |
| 0.5 mM | 3.22 mL | 16.12 mL | 32.25 mL |
| 1 mM | 1.61 mL | 8.06 mL | 16.12 mL |
| 5 mM | 0.32 mL | 1.61 mL | 3.22 mL |
*The above data is based on the productmolecular weight 620.18. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13327 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 2070018-33-4 |
| Formula | C31H30ClN5O3S2 |
| M. Wt | 620.18 |
| Purity | >98% |
| Synonyms | WEHI539 HCl, WEHI 539 HCl |
| SMILES | C1CC2=C(C=C(C=C2)C3=NC(=C(S3)CCCOC4=CC=C(C=C4)CN)C(=O)O)/C(=N/NC5=NC6=CC=CC=C6S5)/C1.Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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WEHI-539 hydrochloride
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