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Biological Activity
WEHI539 is a selective inhibitor of Bcl-XL with IC50 of 1.1 nM.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 17.13 mL | 85.66 mL | 171.32 mL |
| 0.5 mM | 3.43 mL | 17.13 mL | 34.26 mL |
| 1 mM | 1.71 mL | 8.57 mL | 17.13 mL |
| 5 mM | 0.34 mL | 1.71 mL | 3.43 mL |
*The above data is based on the productmolecular weight 583.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13005 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1431866-33-9 |
| Formula | C31H29N5O3S2 |
| M. Wt | 583.72 |
| Purity | >98% |
| Synonyms | WEH I539, WEH-I539 |
| SMILES | OC(C1=C(CCCOC2=CC=C(CN)C=C2)SC(C3=CC4=C(CCC/C4=N\NC5=NC(C=CC=C6)=C6S5)C=C3)=N1)=O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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