Fig. 1 · Structure
Documents & Downloads
Zacopride hydrochloride
5-HT3 Antagonist
Zacopride hydrochloride is a potent 5-HT3 receptor antagonist with a Ki value of 0.38 nM and a 5-HT4 receptor agonist with a Ki value of 373 nM. This compound demonstrates significant biological activities, including modulation of gastrointestinal motility, influence on cardiac function, and the potential to offer anxiolytic and antiemetic effects. Zacopride hydrochloride is primarily utilized in research related to gastrointestinal disorders, cardiovascular conditions, and psychiatric disorders such as anxiety.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 101303-98-4 |
| Applications | 5-HT3 Antagonist |
| Formula | C15H21Cl2N3O2 |
| Molecular Weight | 346.25 |
| SMILES | O=C(NC1CN2CCC1CC2)C3=CC(Cl)=C(N)C=C3OC.[H]Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.