AZD1981

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CRTH2 receptor antagonist

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Catalog No. A13186

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
AZD1981 5mg A13186-5

Regular Price: $60.00

Special Price: $54.00

AZD1981 10mg A13186-10

Regular Price: $100.00

Special Price: $90.00

AZD1981 25mg A13186-25

Regular Price: $200.00

Special Price: $180.00

AZD1981 10mM * 1mL in DMSO A13186-10mM-D

Regular Price: $106.00

Special Price: $95.40

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

AZD1981, as a potent antagonist in a disease relevant cell system, inhibits DK-PGD2-induced CD11b expression in human eosinophils with IC50 of 10 nM.

AZD1981

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Chemical Information

Catalog Num A13186
Actions Antagonist
M. Wt 388.87
Formula C19H17ClN2O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 802904-66-1
Synonyms AZD-1981, AZD 1981
SMILES code CC1=C(C2=C(N1CC(=O)O)C=CC=C2NC(=O)C)SC3=CC=C(C=C3)Cl
Chemical Name 7-Methyl-5-[(3-piperazin-1-ylMethyl)-1,2,4-oxadiazol-5-yl-]-2-[4-(trifluoroMethoxy)benzyl]-2,3-dihydro-1H-isoindol-1-one Methanesulphonat

Biological Activity

Description
AZD1981, as a potent antagonist in a disease relevant cell system, inhibits DK-PGD2-induced CD11b expression in human eosinophils with IC50 of 10 nM.
Targets
CRTh2 (DP2) receptor
4 nM

Solubility

Solubility (25°C)* In vitro DMSO 11 mg/mL (28.28 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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