CC-930 (Tanzisertib)

JNK inhibitor

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Catalog No. A13564

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
CC-930 5mg A13564-5
$180.00
CC-930 10mg A13564-10
$320.00
CC-930 25mg A13564-25
$650.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

CC-930 is kinetically competitive with ATP in the JNK-dependent phosphorylation of the protein substrate c-Jun and potent against all isoforms of JNK (Ki(JNK1) = 44 ± 3 nM, IC50(JNK1) = 61 nM, Ki(JNK2) = 6.2 ± 0.6 nM, IC50(JNK2) = 5 nM, IC50(JNK3) = 5 nM) and selective against MAP kinases ERK1 and p38a with IC50 of 0.48 and 3.4 μM respectively

CC-930 (Tanzisertib)

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Chemical Information

Catalog Num A13564
Actions Inhibitor
M. Wt 448.44
Formula C21H23F3N6O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 899805-25-5
Synonyms Tanzisertib, CC 930, CC930
SMILES code C1COC[[email protected]]1N2C3=NC(=NC=C3N=C2NC4=C(C=C(C=C4F)F)F)NC5CCC(CC5)O
Chemical Name (1S,4r)-4-((9-((S)-tetrahydrofuran-3-yl)-8-((2,4,6-trifluorophenyl)amino)-9H-purin-2-yl)amino)cyclohexanol

Biological Activity

Description
CC-930 is kinetically competitive with ATP in the JNK-dependent phosphorylation of the protein substrate c-Jun and potent against all isoforms of JNK (Ki(JNK1) = 44 ± 3 nM, IC50(JNK1) = 61 nM, Ki(JNK2) = 6.2 ± 0.6 nM, IC50(JNK2) = 5 nM, IC50(JNK3) = 5 nM) and selective against MAP kinases ERK1 and p38a with IC50 of 0.48 and 3.4 μM respectively

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