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|Storage||at -20°C 2 years|
|Synonyms||GF-109203X, GF109203X, GO6850, GO-6850, Bisindolylmaleimide I|
|Chemical Name||2-[1-(3-Dimethylaminopropyl)indol-3?-yl]-3-(indol-3-yl) maleimide|
|GF 109203X is a potent and selective inhibitor of protein kinase C, selective for the α and β1 isoforms (IC50 values are 0.0084, 0.0180, 0.210, 0.132, and 5.8 μM for α, β1, δ, ε and ζ isoforms respectively). Selective over MLCK, PKG and PKA (IC50 values are 0.6, 4.6, and 33 μM respectively). Potent antagonist at the 5-HT3 receptor (Ki = 29.5 nM).|
|Solubility (25°C)*||In vitro||DMSO||82 mg/mL (198.79 mM)|
|Water||<1 mg/mL (<1 mM)|
|Ethanol||<1 mg/mL (<1 mM)|
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
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