GW9508

GPR40 Inhibitor

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Catalog No. A11965

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GW9508 10mg A11965-10
$50.00
GW9508 25mg A11965-25
$100.00
GW9508 50mg A11965-50
$160.00
GW9508 10mM * 1mL in DMSO A11965-10mM-D
$94.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GW 9508 is a cell-permeable aminophenylpropanoate that acts as a potent and selective agonist for the G-protein coupled receptor (GPCR) GRP40/FFA1 receptor (EC50 ?50 nM) with reduced activity towards family members GRP120 (EC50 ?3.5 μM), GRP41/GRP43 (EC50 >50 μM), as well as a panel of eight other free fatty acid (FFA) and prostaglandin receptors.

GW9508

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Chemical Information

Catalog Num A11965
Actions Inhibitor
M. Wt 347.4
Formula C22H21NO3
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 885101-89-3
Synonyms GW 9508, GW-9508
SMILES code C1=CC=C(C=C1)OC2=CC=CC(=C2)CNC3=CC=C(C=C3)CCC(=O)O
Chemical Name 4-[[(3-Phenoxyphenyl)methyl]amino]b?enzenepropanoic acid

Biological Activity

Description
GW 9508 is a cell-permeable aminophenylpropanoate that acts as a potent and selective agonist for the G-protein coupled receptor (GPCR) GRP40/FFA1 receptor (EC50 ?50 nM) with reduced activity towards family members GRP120 (EC50 ?3.5 μM), GRP41/GRP43 (EC50 >50 μM), as well as a panel of eight other free fatty acid (FFA) and prostaglandin receptors.
Targets
GPR40 GPR120
7.32(pEC50)5.46(pEC50)

Solubility

Solubility (25°C)* In vitro DMSO 69 mg/mL (198.61 mM)
Water <1 mg/mL (<1 mM)
Ethanol 69 mg/mL (198.61 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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