OTX015

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BET inhibitor

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Catalog No. A13890

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
OTX015 5mg A13890-5

Regular Price: $70.00

Special Price: $56.00

OTX015 10mg A13890-10

Regular Price: $90.00

Special Price: $72.00

OTX015 25mg A13890-25

Regular Price: $180.00

Special Price: $144.00

OTX015 50mg A13890-50

Regular Price: $250.00

Special Price: $200.00

OTX015 10mM * 1mL in DMSO A13890-10mM-D

Regular Price: $130.00

Special Price: $104.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).

OTX015

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Chemical Information

Catalog Num A13890
Actions Inhibitor
M. Wt 491.99
Formula C25H22ClN5O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 202590-98-5
Synonyms OTX 015, OTX-015
SMILES code CC1=C(SC2=C1C(=N[[email protected]](C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C
Chemical Name (6S)-?4-?(4-?chlorophenyl)-?N-?(4-?hydroxyphenyl)-?2,?3,?9-?trimethyl-?6H-?thieno[3,?2-?f][1,?2,?4]triazolo[4,?3-?a][1,?4]diazepine-?6-?acetamide

Biological Activity

Description
OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Targets
BRDs (Cell-free assay)
10-19 nM(EC50)

Solubility

Solubility (25°C)* In vitro DMSO 98 mg/mL (199.19 mM)
Water <1 mg/mL (<1 mM)
Ethanol 98 mg/mL (199.19 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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