PF-3758309

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PAK4 inhibitor

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Catalog No. A11930

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
PF-3758309 5mg A11930-5

Regular Price: $50.00

Special Price: $42.50

PF-3758309 10mg A11930-10

Regular Price: $80.00

Special Price: $68.00

PF-3758309 25mg A11930-25

Regular Price: $150.00

Special Price: $127.50

PF-3758309 50mg A11930-50

Regular Price: $240.00

Special Price: $204.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.

PF-3758309

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Chemical Information

Catalog Num A11930
Actions Inhibitor
M. Wt 490.2
Formula C25H30N8OS
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 898044-15-0
Synonyms PF-03758309
SMILES code CC1=NC2=C(C(=N1)NC3=NNC4=C3CN(C4(C)C)C(=O)N[[email protected]](CN(C)C)C5=CC=CC=C5)SC=C2
Chemical Name N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]-pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide

Biological Activity

Description
PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.
Targets
Target Value
PAK4IC50: 1.3nM
PAK1ki: 13.7nM
PAK6ki: 17.1nM
PAK5ki: 18.1nM
PAK4ki: 18.7nM
PAK3IC50: 99nM
PAK2IC50: 190nM

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