Fig. 1 · Structure
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(2R,3S)-Azelaprag
Apelin Receptor Agonist
(2R,3S)-Azelaprag is a potent apelin receptor agonist with an EC50 value of 12 nM. This compound serves as a precursor in the study of apelin signaling pathways and their implications in cardiovascular and metabolic research. Its use facilitates the exploration of potential therapeutic applications in conditions related to apelin receptor activation, making it an essential reagent for related biological studies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 2049979-31-7 |
| Applications | Apelin Receptor Agonist |
| Formula | C25H29N7O4S |
| Molecular Weight | 523.61 |
| Synonyms | (2R,3S)-AMG 986 |
| SMILES | O=S(NC1=NN=C(C2=CN=CC(C)=C2)N1C(C(OC)=CC=C3)=C3OC)([C@H](C)[C@H](C4=NC=C(C)C=N4)C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.