5-HT2CR agonist 1 is a selective partial agonist of the 5-HT2C receptor, displaying an effective maximum response (Emax) of 71.09% and an EC50 of 121.5 nM. This compound has been shown to exhibit specificity, with no activity towards 5-HT2A or 5-HT2B receptors. Furthermore, it demonstrates no recruitment activity for β-arrestin and minimal inhibition of hERG channels at 10 μM. This profile makes 5-HT2CR agonist 1 a valuable tool for research in neuropharmacology and receptor signaling pathways.
5-HT2CR agonist 1 is a selective partial agonist of the 5-HT2C receptor, displaying an effective maximum response (Emax) of 71.09% and an EC50 of 121.5 nM. This compound has been shown to exhibit specificity, with no activity towards 5-HT2A or 5-HT2B receptors. Furthermore, it demonstrates no recruitment activity for β-arrestin and minimal inhibition of hERG channels at 10 μM. This profile makes 5-HT2CR agonist 1 a valuable tool for research in neuropharmacology and receptor signaling pathways.
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