5-HT7R antagonist 1

Catalog No.: A60413
G protein-coupled Bile Acid Receptor 1 Antagonist
5-HT7R Antagonist 1 is a G protein-coupled receptor antagonist that selectively inhibits the 5-HT7 receptor, with a Ki value of 6.5 nM. This compound is primarily utilized in research exploring serotonergic signaling pathways and their implications in neuropsychiatric disorders. Its inhibition of 5-HT7R can aid in understanding the receptor's role in various physiological and pathological processes.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Nature Volume 622 Issue 7982 (2023)
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Nature volume 551, pages639-643 (2017)
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Biological Activity
Description5-HT7R Antagonist 1 is a G protein-coupled receptor antagonist that selectively inhibits the 5-HT7 receptor, with a Ki value of 6.5 nM. This compound is primarily utilized in research exploring serotonergic signaling pathways and their implications in neuropsychiatric disorders. Its inhibition of 5-HT7R can aid in understanding the receptor's role in various physiological and pathological processes.
Product Information
Catalog NumA60413
FormulaC14H18Cl2N4
Molecular Weight313.23
CAS Number2759919-13-4
SMILESClC1=CC(C2=NNC=C2N3CCCNCC3)=CC=C1.Cl
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