Target & Activity
| Target | Activity | Value |
|---|---|---|
| mAChR | 0.84 nM(Kb) |
Fig. 1 · Structure
Documents & Downloads
5-hydroxymethyl tolterodine (PNU 200577)
Cat. No.
A11166
CAS
207679-81-0
muscarinic receptor antagonist
5-hydroxymethyl tolterodine is a metabolite of Tolterodine, a muscarinic receptor antagonist used in the treatment of urinary incontinence.
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Biological Activity
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 207679-81-0 |
| Applications | muscarinic receptor antagonist |
| Formula | C22H31NO2 |
| Molecular Weight | 341.49 |
| Synonyms | (R)-5-Hydroxymethyl tolterodine; PNU 200577 |
| SMILES | CC(C)N(CC[C@H](C1=CC=CC=C1)C2=C(C=CC(=C2)CO)O)C(C)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
| Solvent | Reported Solubility |
|---|---|
| DMSO | 60 mg/mL (175.69 mM) |
| Water | Insoluble |
| Ethanol | 60 mg/mL (175.69 mM) |
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.