Fig. 1 · Structure
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ABT-102
Cat. No.
A68763
CAS
808756-71-0
TRPV1 Antagonist
ABT-102 is a potent and highly selective antagonist of the Transient Receptor Potential Vanilloid 1 (TRPV1) channel. This compound effectively elevates heat pain thresholds and diminishes the perception of pain in response to suprathreshold heat stimuli. ABT-102 has demonstrated efficacy in reducing nociceptive responses in various animal models, including those simulating inflammatory pain, bone cancer pain, postoperative pain, and osteoarthritis.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 808756-71-0 |
| Applications | TRPV1 Antagonist |
| Formula | C21H24N4O |
| Molecular Weight | 348.44 |
| SMILES | O=C(NC1=CC=CC2=C1C=NN2)N[C@@H]3CCC4=C3C=CC(C(C)(C)C)=C4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.