Cellular Effect
| Cell Line | Activity | Value | Description | Reference |
|---|---|---|---|---|
| HEK293 | EC50 | 0.21 μM | Partial agonist activity at EGFP-fused human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluorescence assay | [PMID: 22329602] |
| HEK293 | EC50 | 0.45 μM | Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as induction of calcium response by fluorescence assay | [PMID: 22329602] |
| HEK293 | EC50 | 0.72 μM | Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 11 residues expressed in HEK293 cells assessed as induction of calcium response by fluorescence assay | [PMID: 22329602] |
| HEK293 | EC50 | 0.74 μM | Partial agonist activity at human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluorescence assay | [PMID: 22329602] |