AGN 196996

Catalog No.: A16294

RARα antagonist

AGN 196996

AGN 196996 Chemical Structure

CAS NO. 958295-17-5

AGN 196996 is a potent and selective RARα antagonist with Ki value of 2 nM; little binding affinity for RARβ(Ki=1087 nM) and RARγ(Ki=8523 nM).

Availability: In stock

Package Price Qty
5 mg
$320.00
10 mg
$480.00
50 mg
$1,400.00
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Biological Activity

AGN 196996 is a potent and selective RARα antagonist with Ki value of 2 nM; little binding affinity for RARβ(Ki=1087 nM) and RARγ(Ki=8523 nM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.73 mL 103.67 mL 207.33 mL
0.5 mM 4.15 mL 20.73 mL 41.47 mL
1 mM 2.07 mL 10.37 mL 20.73 mL
5 mM 0.41 mL 2.07 mL 4.15 mL

*The above data is based on the productmolecular weight 482.32. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16294
Actions Antagonist
CAS No. 958295-17-5
Formula C24H20BrNO5
M. Wt 482.32
Purity >98%
Synonyms AGN196996, AGN-196996
SMILES CCOC1=C(C=C(C=C1Br)C(=O)NC2=CC=C(C=C2)C(=O)O)C(=O)C3=CC=C(C=C3)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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