Alexidine-d10 is a deuterium-labeled variant of Alexidine, a bis-biguanide compound. It demonstrates significant antifungal and antibiofilm activities against various fungal pathogens. Additionally, Alexidine acts as an anticancer agent by inhibiting the mitochondrial tyrosine phosphatase PTPMT1, leading to mitochondrial apoptosis in mammalian cells. This isotope-labeled version can be particularly useful in studying metabolic pathways and drug interactions in biological systems.
Alexidine-d10 is a deuterium-labeled variant of Alexidine, a bis-biguanide compound. It demonstrates significant antifungal and antibiofilm activities against various fungal pathogens. Additionally, Alexidine acts as an anticancer agent by inhibiting the mitochondrial tyrosine phosphatase PTPMT1, leading to mitochondrial apoptosis in mammalian cells. This isotope-labeled version can be particularly useful in studying metabolic pathways and drug interactions in biological systems.
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